Anastrozole Arimidex for Men: Say Goodbye to Unwanted Estrogen

Here’s one intriguing question that’s probably on your mind right now: why would someone take Anastrozole Arimidex for men? Well, to put it simply, it’s a safe way to reduce elevated estrogen levels.

Most men are not aware that their bodies also produce estrogen, which is traditionally seen as a female hormone. In fact, women and men have both testosterone and estrogen in their bodies; the only difference is the level of each.

Men have higher testosterone levels and women have more estrogen. In men, estradiol is the main biologically active form of estrogen, which is created by the conversion of testosterone.

Estrogen in women regulates the menstrual cycle and affects the reproductive system. In men, it plays such roles as regulating testosterone levels and cholesterol, maintaining libido, and enhancing bone and skin health.

However, as you’d expect, there needs to be a balance between testosterone and estrogen. Otherwise, it can have negative effects on a person’s health.

Older men with a low or borderline-low serum testosterone level can benefit from taking Anastrozole since it increases total and serum bioavailable testosterone to the normal youthful range.

By using pregnenolone cream or pregnenolone supplements, the levels of the compound in the body increases, and this brings about various benefits such as fatigue relief, and delay of the aging process.

On Things to Watch Out For

When the estrogen level in men is too high, it can manifest through the following symptoms:

  • Enlarged breasts (also known as gynecomastia)
  • Feeling fatigued
  • Loss of muscle mass
  • Increase in abdominal fat
  • Sexual dysfunction (erectile dysfunction and decreased libido)
  • Depression and other emotional disturbances
  • Frequent urination, slow urine flow, and symptoms associated with benign prostatic hyperplasia and prostate cancer

One thing to remember is that while estrogen can lower testosterone levels in men, it should not be mistaken for having low testosterone. This is a separate condition with its own set of symptoms.

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What’s Anastrozole for Men?

Anastrozole is a nonsteroidal aromatase inhibitor. This class of drugs inhibits the aromatase enzyme that converts testosterone and other androgen hormones into estrogen hormones.

It’s available under the brand name Arimidex or as a generic drug and is generally given in pill form (taken once daily). It is not an over-the-counter medicine, so you will need a prescription to buy it.

Anastrozole is commonly given to postmenopausal women to stop or slow the development of early-stage breast cancer by decreasing the amount of estrogen they produce.

A doctor may prescribe this medication in addition to radiation, surgery, or chemotherapy to starve these cancers of the estrogen they use. It’s also prescribed in cases of late-stage breast cancer when tamoxifen (brand name Soltamox) no longer works.

In men, Anastrozole is used to reduce the effects of excess testosterone, which can be converted into estrogen by aromatase. It’s most commonly given to men who are undergoing testosterone replacement therapy to prevent the effects of high estradiol levels.

Bodybuilders and other athletes taking anabolic steroids may also take Anastrozole to dodge the side effects of steroid use, although the drug is not approved for this purpose. 

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Risks and Benefits of Anastrozole

Elderly men may particularly benefit from taking Anastrozole. Past the age of 30 or 40, the testosterone produced in the testes gradually declines by around 1% a year.

However, the levels of estradiol continue to remain high due to often increased amounts of fat in middle-age and elderly men, particularly around the abdomen, as well as rising aromatase activity.

In particular, Anastrozole can be effective in cases where low testosterone is due to hypogonadism.

Hypogonadism is a condition in which a problem with the pituitary gland or testicles prevents the body from producing enough testosterone.

This condition is usually treated through hormone replacement therapy to reduce the symptoms of low testosterone. Anastrozole, however, may be a viable alternative to traditional testosterone therapy or treatment.

At the same time, you should consider the long-term effects of taking Anastrozole. For instance, it has been associated with lower bone mineral density, requiring patients with pre-existing osteoporosis to undergo regular monitoring as well as undertaking strategies to protect bone health.

Also while using Anastrozole regular blood tests are needed to confirm you are not taking too much or too little:

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Natural Testosterone Boosters

If, for whatever reason, taking Anastrozole is not appropriate for you, there are several alternatives you can choose for increasing your testosterone levels without resorting to medication.

For one, you could increase your diindolylmethane (DIM) levels. DIM doesn’t actually boost testosterone production but instead ensures that the hormone remains unbound so that the body can use it.

You can increase your DIM levels by eating more cruciferous vegetables, which supplies the body with indole-3-carbinol (I3C) – when broken down, this releases DIM as a byproduct.

Of course, you could also go for natural aromatase inhibitors. Although there are many advantages to laboratory-made estrogen blockers, they can have serious side effects.

This is why it would be better to pursue natural alternatives, such as eating food rich in nutrients that help suppress estrogen and maintain hormonal balance.

Keep in mind that not all supplements made in the laboratory are bad. There are many manufacturers that produce supplements with natural formulations, using plants with known healing properties and naturally occurring compounds as the main ingredients.

For instance, Brassaiopsis Glomerulata is a shrub found in Vietnam whose leaves appear to have bioactive compounds that exhibit aromatase inhibition effects.

Pine Bark Extract is a natural alternative to hormone therapy GnRHa, which stops estrogen production. This herb is not only believed to have similar effects but also reduces erectile dysfunction symptoms.

Before choosing a supplement, make sure that you read the label carefully so you’ll know what ingredients are included in the formulation.

You should also read reviews from trusted sources since they can provide you with important information about the product. But, of course, the best option would always be to visit your doctor before taking a new supplement.

The Bottom Line

While Anastrozole is still the main way to balance hormone levels and increase testosterone, it may not be for everyone. This is why you should explore the various alternatives for boosting natural testosterone production.

While they may take longer to provide the desired outcome, at least you won’t have to worry about suffering from the side effects associated with Anastrozole Arimidex for men.

Alex Eriksson (Research Analysis)

Alex Eriksson is the founder of Anabolic Health, a men’s health blog dedicated to providing honest and research-backed advice for optimal male hormonal health. Anabolic Health aspires to become a trusted resource where men can come and learn how to fix their hormonal problems naturally, without pharmaceuticals.

Ivan Kokhno (Editor)

Ivan is a medical doctor that has five years experience in researching and writing health-related content, SaaS companies, startups, motivation and self-growth resources. He also speak five languages. Therefore, he is able to research any topic five times better than the average writer.

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